SCHEMBL6859720

SCHEMBL6859720

O=C(c1ccco1)c1nc(C(F)(F)F)nc2ccsc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 1.00
ADORA1 P30542 16/20 1.00
APAF1 O14727 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
ADORA2B P29275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6859721 0.81 ADORA2A (0.68) ADORA2AADORA1APAF1NPC1RAB9A
SCHEMBL6214990 0.81 ADORA2A (1.00) ADORA2AADORA1ADORA2B
SCHEMBL6859875 0.80 ADORA2A (1.00) ADORA2AADORA1ADORA2B
SCHEMBL6859683 0.79 ADORA2A (0.65) ADORA2AADORA1NPC1RAB9AKMT2A
SCHEMBL6217242 0.79 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL6858295 0.78 ADORA2A (0.65) ADORA2AADORA1APAF1NPC1RAB9A
SCHEMBL6859469 0.78 ADORA2A (0.72) ADORA2AADORA1ADORA2B
SCHEMBL6853006 0.77 ADORA2A (1.00) ADORA2AADORA1ADORA2B
SCHEMBL6859685 0.77 ADORA2A (0.65) ADORA2AADORA1ADORA2B
SCHEMBL6859939 0.77 ADORA2A (1.00) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787541-B1 MOVEMENT DISORDERS, PARKINSON'S DISEASE VERNALIS RESEARCH LIMITED (GB) 2004-09-07 US disclosed