SCHEMBL6859986

SCHEMBL6859986

O=C1NCN(c2c(Cl)cccc2Cl)c2cc(NC3CCNCC3)cc(-c3ccccc3Cl)c21

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.65
MAPK13 O15264 6/20 0.65
MAPK12 P53778 6/20 0.65
MAPK11 Q15759 6/20 0.65
WEE1 P30291 1/20 0.40
CYP1A2 P05177 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
MEN1 O00255 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703018 0.78 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11
SCHEMBL6696682 0.66 MAPK14 (0.78) MAPK14MAPK13MAPK12MAPK11
SCHEMBL6672308 0.64 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11
SCHEMBL27645212 0.62 TYRO3 (0.43) MAPK14MAPK13MAPK12MAPK11MEN1
SCHEMBL6667987 0.61 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11
SCHEMBL4139369 0.60 HTR6 (0.56) CYP1A2MEN1CYP2D6CYP2C19KMT2A
SCHEMBL83169 0.59 CYP1A2 (0.48) MAPK14MAPK13MAPK12MAPK11CYP1A2
SCHEMBL6668790 0.59 MAPK14 (0.72) MAPK14MAPK13MAPK12MAPK11
SCHEMBL6865000 0.59 MAPK14 (0.76) MAPK14MAPK13MAPK12MAPK11
SCHEMBL918020 0.58 HTR6 (0.49) CYP1A2MEN1KMT2AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6809199-B2 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES MERCK & CO., INC. 2004-10-26 US disclosed