SCHEMBL6860003

SCHEMBL6860003

COc1ccc2c(c1)oc(=O)n2C1CCCC(C(=O)Nc2ccc(-c3ccccc3S(C)(=O)=O)cc2F)C1=O

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 5/20 0.46
FPR1 P21462 4/20 0.46
F10 P00742 15/20 0.45
F2 P00734 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6858734 0.80 F10 (0.65) FPR2FPR1F10
SCHEMBL5950943 0.67 F10 (0.55) FPR2FPR1F10F2
SCHEMBL3830280 0.67 F10 (0.59) FPR2FPR1F10
SCHEMBL7452492 0.66 F10 (0.42) FPR2FPR1F10
SCHEMBL7033131 0.66 F10 (0.63) FPR2FPR1F10
SCHEMBL6258631 0.66 F10 (0.61) FPR2FPR1F10F2
SCHEMBL6853081 0.65 F10 (0.65) FPR2FPR1F10
SCHEMBL6238878 0.65 F10 (0.57) F10F2
SCHEMBL3830204 0.65 F10 (0.81) FPR2FPR1F10
SCHEMBL6859707 0.65 F10 (0.67) FPR2FPR1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030087909-A1 Fused heterocyclic inhibitors of factor Xa BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-05-08 US claimed
US-6790845-B2 HAVING AN ATTACHED NON-AROMATIC HETEROCYCLIC RING BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-09-14 US disclosed
US-20030087909-A1 Fused heterocyclic inhibitors of factor Xa BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030087909-A1 Fused heterocyclic inhibitors of factor Xa TFPI, F11, F12 FPR2 2188/4885FPR1 964/4885F10 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.