SCHEMBL6860760

SCHEMBL6860760

COC(=O)C1CCC(c2nc(NCc3ccc(O)c(OC)c3)c3c(n2)sc2ccccc23)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
SSTR5 P35346 1/20 0.39
ACHE P22303 5/20 0.38
APP P05067 3/20 0.38
BCHE P06276 2/20 0.38
TRPV1 Q8NER1 4/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6859891 0.94 KMT2A (0.40) KMT2AMEN1SSTR5ACHEAPP
SCHEMBL6764725 0.91 PDE10A (0.37) ALDH1A1HSD17B10
SCHEMBL6760546 0.90 PDE5A (0.41)
Bicarbonate SCHEMBL6638242 0.90 PDE5A (0.43) KMT2AMEN1SSTR5ACHEAPP
SCHEMBL6861041 0.89 TRPV1 (0.40) KMT2AMEN1SSTR5ACHEAPP
SCHEMBL6859716 0.88 ESR1 (0.41) KMT2AMEN1ALDH1A1MAPTALOX15
SCHEMBL6764817 0.86 PTPN12 (0.48) KMT2AMEN1KDM4EALDH1A1POLB
Beminafil SCHEMBL6236540 0.84 PDE5A (0.41)
Beminafil SCHEMBL2421274 0.83 PDE5A (0.47)
Beminafil SCHEMBL2421268 0.83 PDE5A (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787548-B1 CARDIOVASCULAR INSUFFICIENCY AND ERECTILE DYSFUNCTION; 3-(4-(3-CHLORO-4-HYDROXYBENZYLAMINO) BENZO(4,5)THIENO(2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2004-09-07 US disclosed