SCHEMBL6861041

SCHEMBL6861041

COc1cc(CNc2nc(C3CCC(CC(=O)O)CC3)nc3sc4ccccc4c23)ccc1O

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.40
ACHE P22303 6/20 0.38
APP P05067 3/20 0.38
BCHE P06276 3/20 0.38
SSTR5 P35346 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6859891 0.91 KMT2A (0.40) TRPV1ACHEAPPBCHESSTR5
SCHEMBL6858279 0.90 PDE5A (0.42)
Bicarbonate SCHEMBL6638242 0.90 PDE5A (0.43) TRPV1ACHEAPPBCHESSTR5
SCHEMBL6860760 0.89 KMT2A (0.40) TRPV1ACHEAPPBCHESSTR5
SCHEMBL6852827 0.88 HSD17B10 (0.39)
SCHEMBL6858238 0.86 PDE5A (0.41)
SCHEMBL7674199 0.85 PDE10A (0.39)
SCHEMBL6859354 0.85 HSD17B10 (0.36)
SCHEMBL7680595 0.84 PDE5A (0.36) KMT2A
SCHEMBL6858363 0.84 PDE5A (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787548-B1 CARDIOVASCULAR INSUFFICIENCY AND ERECTILE DYSFUNCTION; 3-(4-(3-CHLORO-4-HYDROXYBENZYLAMINO) BENZO(4,5)THIENO(2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2004-09-07 US disclosed