SCHEMBL6863442

SCHEMBL6863442

Nc1cccc2[nH]cc(C=O)c12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.64
IMPDH2 P12268 1/20 0.52
PIM1 P11309 2/20 0.40
PIM3 Q86V86 2/20 0.40
PIM2 Q9P1W9 2/20 0.40
CLK1 P49759 1/20 0.39
TRIM24 O15164 1/20 0.39
TRIM33 Q9UPN9 1/20 0.39
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
JAK2 O60674 1/20 0.37
RPS6KA3 P51812 1/20 0.37
MELK Q14680 1/20 0.37
STK24 Q9Y6E0 1/20 0.37
HTR1D P28221 2/20 0.37
HTR1B P28222 1/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29952428 0.82 CYP2A6 (0.70) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL248842 0.79 CYP2A6 (0.66) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29408411 0.79 CYP2A6 (0.66) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29954276 0.78 CYP2A6 (0.64) CYP2A6IMPDH2TRIM24TRIM33HTR1D
SCHEMBL644301 0.78 CYP2A6 (1.00) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29953853 0.78 CYP2A6 (1.00) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL1092485 0.78 CYP2A6 (0.64) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29951940 0.78 CYP2A6 (0.64) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL1337252 0.78 CYP2A6 (0.64) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29935968 0.78 CYP2A6 (0.64) CYP2A6IMPDH2PIM1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed
WO-2011088836-A1 NOVEL 4-(ARYL-4-SULFONYL)-6,6a,7,8,9,10-HEXAHYDRO-4H-4,8,10a-TRIAZA-ACEPHENANTHRYLENE AND 3-ARYLSULFONYL-6,6a,7,8,9,10-HEXAHYDRO-3H-3,8,10a-TRIAZA-CYCLOPENTA[C]FLUORENE DERIVATIVES AS SEROTONIN 5-HT6 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed