SCHEMBL6863535

SCHEMBL6863535

O=C(CN1CCN(Cc2ccccc2)CC1)NO

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.68
MEN1 O00255 3/20 0.68
ATM Q13315 1/20 0.65
HDAC4 P56524 1/20 0.65
KCNH2 Q12809 1/20 0.65
HDAC1 Q13547 1/20 0.65
ALDH1A1 P00352 9/20 0.64
KDM4E B2RXH2 1/20 0.63
MAPT P10636 2/20 0.62
GAA P10253 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
LMNA P02545 1/20 0.62
SIGMAR1 Q99720 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
MAPK1 P28482 1/20 0.60
CYP2C19 P33261 1/20 0.60
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA7 P43166 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31122768 0.85 ALDH1A1 (0.68) KMT2AMEN1HDAC4KCNH2HDAC1
SCHEMBL10041823 0.85 ALDH1A1 (0.64) KMT2AMEN1ATMALDH1A1KDM4E
SCHEMBL4084709 0.85 KMT2A (0.73) KMT2AMEN1ATMALDH1A1KDM4E
SCHEMBL4818022 0.84 CA1 (0.76) KMT2AMEN1ATMALDH1A1KDM4E
SCHEMBL12150889 0.84 KMT2A (0.76) KMT2AMEN1HDAC4KCNH2HDAC1
SCHEMBL31122730 0.83 KMT2A (0.57) KMT2AMEN1ATMHDAC4KCNH2
SCHEMBL31122711 0.83 HDAC1 (0.57) KMT2AMEN1HDAC4KCNH2HDAC1
SCHEMBL2717435 0.82 ALDH1A1 (0.72) KMT2AMEN1ATMHDAC4KCNH2
SCHEMBL8033956 0.82 ALDH1A1 (0.72) KMT2AMEN1ATMHDAC4KCNH2
SCHEMBL21044023 0.82 ALDH1A1 (0.72) KMT2AMEN1ATMHDAC4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed
WO-1998005332-A1 NOVEL HETEROCYCLE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-12 WO disclosed