SCHEMBL6864121

SCHEMBL6864121

COc1ccc(CC(=O)O)c(Oc2cccc(N)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.56
CAMK2A Q9UQM7 2/20 0.52
ALDH1A1 P00352 1/20 0.51
CYP3A4 P08684 1/20 0.51
KDM4E B2RXH2 3/20 0.49
POLB P06746 1/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 1/20 0.43
MAOB P27338 1/20 0.43
PTGS1 P23219 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
TSPO P30536 3/20 0.42
SLC1A5 Q15758 1/20 0.42
LCK P06239 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6175515 0.86 CAMK2A (0.68) HSD17B10CAMK2AALDH1A1KDM4EPOLB
SCHEMBL6865044 0.81 HSD17B10 (0.51) HSD17B10CAMK2AALDH1A1KDM4EPOLB
SCHEMBL11577618 0.80 HSD17B10 (0.63) HSD17B10CAMK2AKDM4EPOLBSMN1; SMN2
SCHEMBL9152146 0.80 SLC1A5 (0.57) HSD17B10CAMK2AKDM4EPOLBPTGDR2
SCHEMBL1097902 0.79 HSD17B10 (0.75) HSD17B10ALDH1A1KDM4EPOLBPTGS1
SCHEMBL30831943 0.79 HSD17B10 (0.75) HSD17B10ALDH1A1KDM4EPOLBPTGS1
SCHEMBL9148385 0.79 SLC1A5 (0.56) HSD17B10CAMK2AKDM4EPOLBPTGDR2
Hydrochloric Acid SCHEMBL2527027 0.77 HSD17B10 (0.73) HSD17B10ALDH1A1KDM4EPOLBPTGS1
SCHEMBL6179348 0.76 CAMK2A (0.54) HSD17B10CAMK2AALDH1A1KDM4EPOLB
Acetic Acid SCHEMBL4630447 0.75 CYP3A4 (0.77) ALDH1A1CYP3A4KDM4EPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed