SCHEMBL6864586

SCHEMBL6864586

CC(C)N1CCCN(c2nc3c(OC(N)=O)cccc3[nH]2)CC1

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.45
PARP2 Q9UGN5 1/20 0.43
NPY5R Q15761 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869126 0.96 PARP1 (0.48) PARP1PARP2NPY5R
SCHEMBL6873048 0.86 PARP1 (0.47) PARP1NPY5R
SCHEMBL7417491 0.86 NPY5R (0.45) PARP1PARP2NPY5R
SCHEMBL6584369 0.85 PARP1 (0.50) PARP1PARP2
SCHEMBL6873874 0.84 PARP1 (0.46) PARP1NPY5R
SCHEMBL5620810 0.84 PARP1 (0.64) PARP1PARP2
SCHEMBL6874969 0.84 PARP1 (0.51) PARP1NPY5R
SCHEMBL6873342 0.82 PARP1 (0.46) PARP1PARP2
SCHEMBL6864630 0.82 PARP1 (0.49) PARP1NPY5R
SCHEMBL6864445 0.81 PARP1 (0.46) PARP1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed