SCHEMBL6864630

SCHEMBL6864630

CC(=O)N1CCN(c2nc3c(OC(N)=O)cccc3[nH]2)CC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.49
NAMPT P43490 1/20 0.42
NPY5R Q15761 1/20 0.42
HTR2B P41595 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873874 0.96 PARP1 (0.46) PARP1NAMPTNPY5RHTR2B
SCHEMBL6874969 0.88 PARP1 (0.51) PARP1NPY5R
SCHEMBL7409990 0.86 PARP1 (0.43) PARP1NAMPTNPY5RHTR2B
SCHEMBL6869126 0.85 PARP1 (0.48) PARP1NPY5R
SCHEMBL6869623 0.85 PARP1 (0.49) PARP1NAMPTNPY5R
SCHEMBL6873048 0.84 PARP1 (0.47) PARP1NPY5R
SCHEMBL6869369 0.84 PARP1 (0.49) PARP1NPY5R
SCHEMBL5621895 0.82 PARP1 (0.71) PARP1
SCHEMBL6864586 0.82 PARP1 (0.45) PARP1NPY5R
SCHEMBL6864445 0.81 PARP1 (0.46) PARP1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed