SCHEMBL6865040

SCHEMBL6865040

COCCNC(=O)c1c(C)nn(-c2cccc3cc(Cc4cc(F)cc(Cl)c4)sc23)c1C

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 14/20 0.72
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TP53 P04637 2/20 0.37
DGAT2 Q96PD7 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13505899 0.92 GPR52 (0.71) GPR52NPC1RAB9A
SCHEMBL13506218 0.88 GPR52 (0.57) GPR52NPC1RAB9ATP53
SCHEMBL6865110 0.86 GPR52 (0.76) GPR52NPC1RAB9A
SCHEMBL13505722 0.86 GPR52 (0.53) GPR52KMT2A
SCHEMBL13505947 0.85 PDE4B (0.52) GPR52KMT2A
SCHEMBL6865361 0.84 GPR52 (0.73) GPR52NPC1RAB9ATP53
SCHEMBL13505642 0.83 GPR52 (1.00) GPR52
SCHEMBL6864696 0.82 GPR52 (0.61) GPR52NPC1RAB9A
SCHEMBL13506568 0.80 GPR52 (0.54) GPR52NPC1RAB9ATP53
SCHEMBL6863956 0.80 GPR52 (0.71) GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2518054-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2012-10-31 EP disclosed
WO-2011078360-A1 AMIDE COMPOUND 武田薬品工業株式会社 (JP) 2011-06-30 WO disclosed