SCHEMBL6866552

SCHEMBL6866552

CC(=O)OC(C(=O)N[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.57
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.41
MAPK8 P45983 3/20 0.41
CYP2C9 P11712 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
MAPK14 Q16539 1/20 0.41
MCHR1 Q99705 6/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADRA2A P08913 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6866555 1.00 TSHR (0.57) TSHRMAPK1ALDH1A1GAAHPGD
SCHEMBL6867727 0.90 TSHR (0.43) TSHRALDH1A1GAAHPGDMAPK8
SCHEMBL6457914 0.86 CCR1 (0.43) MAPK8CYP2C9CCNE1CDK2MAPK9
SCHEMBL6457922 0.86 CCR1 (0.43) MAPK8CYP2C9CCNE1CDK2MAPK9
SCHEMBL6880601 0.82 LMNA (0.41) GAALMNAMAPK8CYP2C9CCNE1
SCHEMBL6880608 0.82 LMNA (0.41) GAALMNAMAPK8CYP2C9CCNE1
SCHEMBL6877430 0.81 MAPK8 (0.41) MAPK8CYP2C9CCNE1CDK2MAPK9
SCHEMBL6877427 0.81 MAPK8 (0.41) MAPK8CYP2C9CCNE1CDK2MAPK9
SCHEMBL6879679 0.80 TSHR (0.47) TSHRMAPK1HPGDMAPK8CYP2C9
SCHEMBL6879696 0.80 TSHR (0.47) TSHRMAPK1HPGDMAPK8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed