SCHEMBL6867345

SCHEMBL6867345

CC1CCCN(C(=O)c2cc(N)n3nc(-c4nccs4)nc3c2)C1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.63
RECQL P46063 1/20 0.46
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871877 0.89 ADORA2A (0.48) ADORA2AALDH1A1
SCHEMBL6870280 0.89 ADORA2A (0.53) ADORA2AALDH1A1HPGD
SCHEMBL6863814 0.87 ADORA2A (0.67) ADORA2AHPGD
SCHEMBL6870030 0.86 ADORA2A (0.66) ADORA2AHPGD
SCHEMBL6863267 0.86 ADORA2A (0.66) ADORA2AHPGD
SCHEMBL6863682 0.86 ADORA2A (0.66) ADORA2AHPGD
SCHEMBL6872157 0.85 ADORA2A (0.50) ADORA2A
SCHEMBL6867753 0.85 ADORA2A (0.61) ADORA2AALDH1A1HPGD
SCHEMBL6870718 0.85 ADORA2A (0.67) ADORA2AALDH1A1HPGD
SCHEMBL6863359 0.83 ADORA2A (0.47) ADORA2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed