SCHEMBL686756

SCHEMBL686756

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2cccn(Cc3cc(F)ccc3Br)c2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
KDM4E B2RXH2 8/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
HPGD P15428 3/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGER3 P43115 11/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPK1 P28482 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
CTSA P10619 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688001 0.91 KDM4E (0.48) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL687966 0.90 ALDH1A1 (0.46) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL686797 0.90 KDM4E (0.48) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL27587259 0.89 ALDH1A1 (0.55) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL686984 0.89 ALDH1A1 (0.55) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL688388 0.88 PTGER3 (0.48) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL688009 0.88 PTGER3 (0.58) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL687142 0.87 MAPT (0.44) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL688469 0.87 KDM4E (0.58) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL688211 0.86 PTGER3 (0.46) ALDH1A1KDM4EMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1176956-B1 CARBOXYLIC ACID DERIVATIVES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed