SCHEMBL6869279

SCHEMBL6869279

CN(C)c1ccnc(NC2CCC(NC(=O)Nc3ccccc3Cl)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
EPHX2 P34913 1/20 0.47
MCHR1 Q99705 5/20 0.45
ADRA2A P08913 3/20 0.45
HRH1 P35367 3/20 0.45
HTR2B P41595 3/20 0.45
PAK1 Q13153 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADRA1A P35348 2/20 0.44
DRD2 P14416 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1B P35368 1/20 0.43
MAPK3 P27361 1/20 0.43
MAPK1 P28482 1/20 0.43
MAPK8 P45983 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869275 1.00 MAPK14 (0.54) MAPK14NPC1RAB9AEPHX2MCHR1
SCHEMBL6876089 0.91 TSHR (0.57) MAPK14NPC1RAB9AEPHX2MCHR1
SCHEMBL6876093 0.91 TSHR (0.57) MAPK14NPC1RAB9AEPHX2MCHR1
Hydrochloric Acid SCHEMBL6460685 0.91 MAPK14 (0.45) MAPK14NPC1RAB9AMCHR1ADRA2A
Hydrochloric Acid SCHEMBL6460688 0.91 MAPK14 (0.45) MAPK14NPC1RAB9AMCHR1ADRA2A
SCHEMBL6872847 0.89 EPHX2 (0.47) MAPK14EPHX2MCHR1ADRA2AHRH1
SCHEMBL6872853 0.89 EPHX2 (0.47) MAPK14EPHX2MCHR1ADRA2AHRH1
SCHEMBL6880649 0.88 AURKB (0.41) MAPK14MCHR1ADRA2AHRH1HTR2B
SCHEMBL6878450 0.88 MAPK8 (0.41) MAPK14MCHR1ADRA2AHRH1HTR2B
SCHEMBL6878449 0.88 MAPK8 (0.41) MAPK14MCHR1ADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed