SCHEMBL6869334

SCHEMBL6869334

CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)c1nc(COS(C)(=O)=O)ncc1-c1ccccc1Cl

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.57
GPBAR1 Q8TDU6 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696891 0.81 TACR1 (0.56) TACR1GPBAR1
SCHEMBL6016333 0.79 TACR1 (0.56) TACR1
SCHEMBL5779622 0.76 TACR1 (0.75) TACR1GPBAR1
SCHEMBL7702182 0.75 TACR1 (0.60) TACR1
SCHEMBL5782663 0.74 TACR1 (0.72) TACR1GPBAR1
SCHEMBL5966350 0.74 TACR1 (0.80) TACR1GPBAR1
SCHEMBL6862193 0.74 TACR1 (0.80) TACR1GPBAR1
Hydrochloric Acid SCHEMBL6869633 0.73 TACR1 (0.78) TACR1GPBAR1
SCHEMBL6862358 0.71 TACR1 (0.72) TACR1
SCHEMBL6869431 0.70 TACR1 (0.52) TACR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187814-B1 5-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-18 EP disclosed
US-6756380-B1 NEUROKININ 1 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. 2004-06-29 US disclosed
EP-1187814-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
WO-2000073278-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed