SCHEMBL6869442

SCHEMBL6869442

NC(=O)Oc1cccc2[nH]c(N3CCCN(Cc4ccccc4)CC3)nc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.47
KDR P35968 1/20 0.47
AURKB Q96GD4 1/20 0.47
PARP1 P09874 9/20 0.45
TSHR P16473 2/20 0.44
HTT P42858 1/20 0.44
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
DRD3 P35462 2/20 0.44
GAA P10253 1/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ATM Q13315 1/20 0.43
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873471 0.96 AURKA (0.49) AURKAKDRAURKBPARP1TSHR
SCHEMBL7413218 0.92 TSHR (0.46) AURKAKDRAURKBPARP1TSHR
SCHEMBL6580774 0.86 PARP1 (0.56) AURKAKDRAURKBPARP1
SCHEMBL6873342 0.85 PARP1 (0.46) AURKAAURKBPARP1
SCHEMBL5620780 0.85 AURKA (0.62) AURKAKDRAURKBPARP1
SCHEMBL6864807 0.84 PARP1 (0.40) PARP1DRD2DRD3
SCHEMBL6872540 0.83 PARP1 (0.39) PARP1
SCHEMBL6869630 0.83 PARP1 (0.41) PARP1
SCHEMBL6870125 0.83 PARP1 (0.44) PARP1
SCHEMBL6590662 0.83 AURKB (0.72) AURKAKDRAURKBPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed