SCHEMBL6869630

SCHEMBL6869630

NC(=O)Oc1cccc2[nH]c(N3CCCN(CCc4ccc(O)cc4)CC3)nc12

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.41
HRH1 P35367 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
CYP3A4 P08684 1/20 0.36
ABCC1 P33527 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871167 0.96 PARP1 (0.43) PARP1CYP3A4ABCC1
SCHEMBL6870125 0.93 PARP1 (0.44) PARP1CYP3A4ABCC1
SCHEMBL6870272 0.92 PARP1 (0.40) PARP1HRH1HRH3CYP3A4ABCC1
SCHEMBL6871574 0.92 PARP1 (0.40) PARP1HRH1HRH3CYP3A4ABCC1
SCHEMBL6869177 0.92 PARP1 (0.41) PARP1HRH3
SCHEMBL6864807 0.92 PARP1 (0.40) PARP1HRH1CYP3A4ABCC1
SCHEMBL6871608 0.91 PARP1 (0.47) PARP1HRH1HRH3KCNH2
SCHEMBL7043428 0.90 PARP1 (0.41) PARP1CYP3A4ABCC1
SCHEMBL6864914 0.90 PARP1 (0.41) PARP1CYP3A4
SCHEMBL6875539 0.90 PARP1 (0.39) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed