SCHEMBL6869604

SCHEMBL6869604

CC1C=CC(C)N1C(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.69
F12 P00748 11/20 0.45
F2 P00734 9/20 0.45
PLAU P00749 2/20 0.44
PLG P00747 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867942 0.83 ADORA2A (0.71) ADORA2AF12F2PLAUPLG
SCHEMBL6867372 0.82 ADORA2A (0.74) ADORA2AF12F2PLAUPLG
SCHEMBL6869818 0.82 ADORA2A (0.70) ADORA2AF12F2PLAUPLG
SCHEMBL6867568 0.81 ADORA2A (1.00) ADORA2AF12F2PLAUPLG
SCHEMBL6871685 0.81 ADORA2A (0.80) ADORA2AF12F2PLAUPLG
SCHEMBL6867379 0.81 ADORA2A (0.66) ADORA2AF12F2PLAUPLG
SCHEMBL6863273 0.81 ADORA2A (0.71) ADORA2AF12F2
SCHEMBL6871467 0.80 ADORA2A (0.98) ADORA2AF12F2PLAU
SCHEMBL6869099 0.80 ADORA2A (0.98) ADORA2AF12F2PLAU
SCHEMBL6869091 0.80 ADORA2A (0.98) ADORA2AF12F2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed