SCHEMBL6869099

SCHEMBL6869099

Nc1cc(C(=O)N2CCCCC2)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.98

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.98
HPGD P15428 2/20 0.51
CYP2C9 P11712 1/20 0.47
F2 P00734 2/20 0.43
F12 P00748 2/20 0.43
PLAU P00749 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869091 1.00 ADORA2A (0.98) ADORA2AHPGDCYP2C9F2F12
SCHEMBL6871467 1.00 ADORA2A (0.98) ADORA2AHPGDCYP2C9F2F12
SCHEMBL6867568 0.99 ADORA2A (1.00) ADORA2AHPGDCYP2C9F2F12
SCHEMBL6871685 0.88 ADORA2A (0.80) ADORA2AF2F12PLAU
SCHEMBL7143076 0.87 ADORA2A (0.78) ADORA2AHPGD
SCHEMBL6873970 0.85 ADORA2A (0.74) ADORA2AHPGD
SCHEMBL6867372 0.84 ADORA2A (0.74) ADORA2AF2F12PLAU
SCHEMBL6867145 0.84 ADORA2A (0.71) ADORA2AHPGD
SCHEMBL6863643 0.84 ADORA2A (0.73) ADORA2AHPGD
SCHEMBL6868104 0.83 ADORA2A (0.72) ADORA2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed