SCHEMBL7043428

SCHEMBL7043428

COC(=O)c1ccc(CCN2CCCN(c3nc4c(OC(N)=O)cccc4[nH]3)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.41
ABCC1 P33527 2/20 0.40
CYP3A4 P08684 1/20 0.40
DRD2 P14416 3/20 0.40
DRD4 P21917 3/20 0.40
DRD3 P35462 3/20 0.40
CHKA P35790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875504 0.97 PARP1 (0.43) PARP1ABCC1CYP3A4
SCHEMBL6871608 0.91 PARP1 (0.47) PARP1DRD2
SCHEMBL6869177 0.91 PARP1 (0.41) PARP1
SCHEMBL6869630 0.90 PARP1 (0.41) PARP1ABCC1CYP3A4
SCHEMBL6870125 0.90 PARP1 (0.44) PARP1ABCC1CYP3A4
SCHEMBL6864807 0.89 PARP1 (0.40) PARP1ABCC1CYP3A4DRD2DRD3
SCHEMBL6871574 0.89 PARP1 (0.40) PARP1ABCC1CYP3A4
SCHEMBL6870272 0.89 PARP1 (0.40) PARP1ABCC1CYP3A4
SCHEMBL6875539 0.88 PARP1 (0.39) PARP1DRD2DRD4DRD3
SCHEMBL5621202 0.88 PARP1 (0.54) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed