SCHEMBL6870562

SCHEMBL6870562

CCN(CCOC)C(=O)c1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.48
MLYCD O95822 1/20 0.37
PDE11A Q9HCR9 1/20 0.37
CRHR1 P34998 1/20 0.35
ADORA2B P29275 2/20 0.33
ADORA1 P30542 2/20 0.33
CNR2 P34972 1/20 0.33
NAMPT P43490 1/20 0.33
F2 P00734 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868365 0.95 ADORA2A (0.44) ADORA2APDE11ACRHR1ADORA2BADORA1
SCHEMBL6863143 0.90 ADORA2A (0.58) ADORA2APDE11AADORA2BADORA1
SCHEMBL6871315 0.89 ADORA2A (0.50) ADORA2APDE11ACRHR1
SCHEMBL6867673 0.86 ADORA2A (0.48) ADORA2APDE11AADORA2BADORA1F2
SCHEMBL6870319 0.83 ADORA2A (0.49) ADORA2APDE11AADORA2BADORA1
SCHEMBL6869063 0.83 ADORA2A (0.46) ADORA2APDE11AADORA2BADORA1F2
SCHEMBL6867506 0.83 ADORA2A (0.50) ADORA2APDE11AF2
SCHEMBL6870657 0.83 ADORA2A (0.50) ADORA2APDE11AF2
SCHEMBL6866988 0.82 ADORA2A (0.60) ADORA2APDE11AADORA2BADORA1
SCHEMBL6873639 0.82 ADORA2A (0.46) ADORA2APDE11AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed