SCHEMBL6870765

SCHEMBL6870765

Bc1nc(Cl)ccc1NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.44
LCK P06239 2/20 0.41
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
CYP17A1 P05093 2/20 0.39
MAPKAPK2 P49137 2/20 0.39
PSMB8 P28062 1/20 0.39
METAP1 P53582 1/20 0.39
P2RX7 Q99572 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
ELANE P08246 1/20 0.37
CTRB1 P17538 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074732 0.86 ATR (0.48) ATRLCKKMT2ALMNACYP17A1
SCHEMBL12133550 0.84 LCK (0.46) ATRLCKKMT2ALMNACYP17A1
SCHEMBL15951249 0.83 ATR (0.43) ATRLCKKMT2ALMNACYP17A1
SCHEMBL16533461 0.83 ATR (0.43) ATRLCKKMT2ALMNACYP17A1
SCHEMBL19384200 0.81 XPO1 (0.44) ATRLCKKMT2ALMNACYP17A1
SCHEMBL3710643 0.81 MAPKAPK2 (0.45) ATRLCKKMT2ALMNACYP17A1
SCHEMBL12133539 0.81 ATR (0.44) ATRLCKKMT2ALMNACYP17A1
SCHEMBL25028777 0.80 METAP1 (0.44) ATRLCKKMT2ALMNACYP17A1
SCHEMBL31120609 0.80 LCK (0.43) ATRLCKKMT2ALMNACYP17A1
SCHEMBL29439638 0.80 METAP1 (0.41) ATRLCKKMT2ALMNACYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119694-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed