SCHEMBL16533461

SCHEMBL16533461

CC(C)(C)OC(=O)Nc1ccc(Cl)nc1Br

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.43
LCK P06239 3/20 0.40
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
MAPKAPK2 P49137 2/20 0.39
CYP17A1 P05093 2/20 0.39
METAP1 P53582 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
P2RX7 Q99572 1/20 0.38
BRD9 Q9H8M2 1/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074732 0.84 ATR (0.48) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL12133550 0.83 LCK (0.46) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL6870765 0.83 ATR (0.44) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL31438981 0.82 ATR (0.39) ATRLCKKMT2ACYP17A1METAP1
SCHEMBL26944256 0.82 ATR (0.39) ATRLCKKMT2ACYP17A1METAP1
SCHEMBL15951249 0.82 ATR (0.43) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL25271015 0.81 ATR (0.45) ATRLCKMAPKAPK2CYP17A1METAP1
SCHEMBL3710643 0.79 MAPKAPK2 (0.45) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL12133539 0.79 ATR (0.44) ATRLCKKMT2ALMNAMAPKAPK2
SCHEMBL19384200 0.79 XPO1 (0.44) ATRLCKKMT2ALMNAMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12617789-B2 Small molecular inhibitors of NF-κb inducing kinase JANSSEN PHARMACEUTICA NV (BE) 2026-05-05 US disclosed
US-12509431-B2 1,4-dihydroquinazolinone compounds and uses thereof EDGEWISE THERAPEUTICS, INC. (US) 2025-12-30 US disclosed
US-20250361213-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS INC (US) 2025-11-27 US disclosed
EP-4594307-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2025-08-06 EP disclosed
US-20250154111-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. 2025-05-15 US disclosed
US-20250034141-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2025-01-30 US disclosed
EP-4467199-A2 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2024-11-27 EP disclosed
US-12152027-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-11-26 US disclosed
WO-2024206347-A1 FUSED THIADIAZINE DIOXIDE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2024-10-03 WO disclosed
EP-3976597-B1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2024-08-28 EP disclosed
US-20220089595-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2022-03-24 US disclosed
US-11254673-B2 Small molecule inhibitors of NF-κB inducing kinase JANSSEN PHARMACEUTICA NV (BE) 2022-02-22 US disclosed
US-20220048916-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-02-17 US disclosed
US-11230545-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-01-25 US disclosed
US-20210332045-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-10-28 US disclosed
EP-3888652-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-10-06 EP disclosed
US-20180065932-A1 ANTIVIRAL COMPOUNDS ALIOS BIOPHARMA, INC. 2018-03-08 US disclosed
US-20150065504-A1 ANTIVIRAL COMPOUNDS ALIOS BIOPHARMA, INC. 2015-03-05 US disclosed
US-20150065504-A1 ANTIVIRAL COMPOUNDS ALIOS BIOPHARMA, INC. 2015-03-05 US disclosed
WO-2015026792-A1 ANTIVIRAL COMPOUNDS ALIOS BIOPHARMA, INC. (US) 2015-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220089595-A1 HETEROCYCLIC COMPOUND MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885
US-20250034141-A1 HETEROCYCLIC COMPOUND MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885
US-11230545-B2 Heterocyclic compound MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885
US-12509431-B2 1,4-dihydroquinazolinone compounds and uses thereof TNNT2, TNNI3, TNNC1 ATR 3085/4885LCK 4097/4885KMT2A 3822/4885
US-20180065932-A1 ANTIVIRAL COMPOUNDS MAVS, SARS1, ZC3HAV1 ATR 1930/4885LCK 3440/4885KMT2A 4241/4885
US-20150065504-A1 ANTIVIRAL COMPOUNDS MAVS, SARS1, ZC3HAV1 ATR 1930/4885LCK 3440/4885KMT2A 4241/4885
US-20210332045-A1 HETEROCYCLIC COMPOUND MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885
US-11254673-B2 Small molecule inhibitors of NF-κB inducing kinase NFKBIA, IKBKB, CHUK ATR 3528/4885LCK 75/4885KMT2A 1080/4885
US-20250154111-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF TNNI3, TNNT2, SDHA ATR 4439/4885LCK 3768/4885KMT2A 3454/4885
US-12617789-B2 Small molecular inhibitors of NF-κb inducing kinase IRAK3, IKBKB, IKBKG ATR 3093/4885LCK 141/4885KMT2A 2492/4885
US-12152027-B2 Heterocyclic compound MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885
US-20250361213-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF TNNI3, TNNT2, SDHA ATR 4439/4885LCK 3768/4885KMT2A 3454/4885
US-20220048916-A1 HETEROCYCLIC COMPOUND MALT1, SQSTM1, PPM1D ATR 3457/4885LCK 1446/4885KMT2A 2085/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.