SCHEMBL687265

SCHEMBL687265

CCOc1cccc(Cl)c1Cn1cc(C)c(O)c(NC(=O)N[C@@H](CC(=O)O)c2cccc(C(F)(F)F)c2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 8/20 0.40
WDR5 P61964 2/20 0.39
IL1B P01584 1/20 0.37
P2RX7 Q99572 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
HTT P42858 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
FFAR1 O14842 1/20 0.34
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688105 0.91 ITGB3 (0.39) CTSAWDR5P2RX7SMN1; SMN2ALDH1A1
SCHEMBL686989 0.91 SMN1; SMN2 (0.38) CTSASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL687802 0.90 CTSA (0.34) CTSAWDR5P2RX7SMN1; SMN2ALDH1A1
SCHEMBL687119 0.89 SMN1; SMN2 (0.36) SMN1; SMN2ALDH1A1HTTKMT2AKDM4E
SCHEMBL688507 0.88 SMN1; SMN2 (0.38) CTSASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL687715 0.88 CTSA (0.39) CTSASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL688386 0.87 SMN1; SMN2 (0.40) CTSASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL687688 0.87 SMN1; SMN2 (0.37) CTSASMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL687907 0.87 SMN1; SMN2 (0.38) CTSAP2RX7SMN1; SMN2ALDH1A1KMT2A
SCHEMBL688501 0.86 SMN1; SMN2 (0.40) CTSAP2RX7SMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed