SCHEMBL6873248

SCHEMBL6873248

COc1nc(NC2CCC(NC(=O)c3cc(Cl)cc(Cl)c3)CC2)ncc1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 13/20 0.57
ADRA2A P08913 6/20 0.57
HRH1 P35367 6/20 0.57
HTR2B P41595 6/20 0.57
ADRA1A P35348 3/20 0.50
CNR1 P21554 1/20 0.47
KCNH2 Q12809 1/20 0.47
AURKB Q96GD4 1/20 0.47
HPGDS O60760 1/20 0.45
LRRK2 Q5S007 1/20 0.44
CCNA2 P20248 2/20 0.44
CDK2 P24941 2/20 0.44
BRD4 O60885 2/20 0.43
CHEK1 O14757 1/20 0.42
IKBKB O14920 1/20 0.42
AURKA O14965 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
CHEK2 O96017 1/20 0.42
ABL1 P00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873245 1.00 MCHR1 (0.57) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6878288 0.89 MCHR1 (0.71) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6878285 0.89 MCHR1 (0.71) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6461744 0.87 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6461733 0.87 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6875281 0.85 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6875276 0.85 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6458198 0.83 MCHR1 (0.81) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6458207 0.83 MCHR1 (0.81) MCHR1ADRA2AHRH1HTR2BADRA1A
Hydrochloric Acid SCHEMBL6462069 0.82 MCHR1 (0.79) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed