SCHEMBL6873370

SCHEMBL6873370

CN(C)c1ccnc(N[C@H]2CC[C@@H](NC(=O)c3ccccc3-c3ccccc3)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MCHR1 Q99705 14/20 0.48
MAPK8 P45983 2/20 0.46
MAPK14 Q16539 1/20 0.46
ADRA2A P08913 7/20 0.44
HRH1 P35367 5/20 0.44
HTR2B P41595 5/20 0.44
ADRA1A P35348 3/20 0.44
CNR1 P21554 1/20 0.41
KCNH2 Q12809 1/20 0.41
AURKB Q96GD4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873378 1.00 GAA (0.54) GAAMEN1KMT2AALDH1A1LMNA
SCHEMBL6878850 0.85 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6878847 0.85 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6456005 0.85 KLK7 (0.59) GAAMEN1KMT2AALDH1A1LMNA
SCHEMBL6456016 0.85 KLK7 (0.59) GAAMEN1KMT2AALDH1A1LMNA
SCHEMBL6877485 0.84 MCHR1 (0.52) KMT2AMCHR1ADRA2AHRH1HTR2B
SCHEMBL6877476 0.84 MCHR1 (0.52) KMT2AMCHR1ADRA2AHRH1HTR2B
SCHEMBL6874303 0.84 TSHR (0.46) GAAMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL6874310 0.84 TSHR (0.46) GAAMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL6879228 0.83 MCHR1 (0.46) MCHR1MAPK8ADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed