SCHEMBL687401

SCHEMBL687401

CCNC(=O)Nc1cc[c]cc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
NPC1 O15118 1/20 0.44
THRB P10828 1/20 0.44
RAB9A P51151 1/20 0.44
NOX1 Q9Y5S8 1/20 0.44
EPHX2 P34913 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 2/20 0.40
LMNA P02545 1/20 0.37
MAPT P10636 2/20 0.37
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7107830 0.85 ALDH1A1 (0.44) POLBMAPK1KMT2AMEN1KDM4E
SCHEMBL5217967 0.84 KMT2A (0.42) POLBMAPK1KMT2AMEN1KDM4E
SCHEMBL687471 0.81 POLB (0.47) POLBMAPK1KMT2AMEN1KDM4E
SCHEMBL2989161 0.80 CYP1A2 (0.47) POLBKMT2AMEN1KDM4EALDH1A1
SCHEMBL7113819 0.78 MAPT (0.37) POLBMAPK1KMT2AMEN1KDM4E
SCHEMBL13480579 0.78 POLB (0.68) POLBMAPK1KMT2AMEN1KDM4E
SCHEMBL7110018 0.78 PDE3B (0.36) TSHRLMNA
SCHEMBL1901639 0.77 KDM4E (0.52) KMT2AMEN1KDM4EALDH1A1GAA
SCHEMBL27678713 0.77 GAA (0.41) POLBKMT2AMEN1KDM4ENPC1
SCHEMBL1355211 0.73 KMT2A (0.52) KMT2AMEN1KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667966-B1 N-ALKYLATED DIAMINOPROPANE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-02-29 EP disclosed