SCHEMBL6874447

SCHEMBL6874447

CN(C)c1cc(NC2CCC(NC(=S)Nc3ccc4c(c3)OCCO4)CC2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.47
ALDH1A1 P00352 5/20 0.44
MAPT P10636 7/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
ALOX12 P18054 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
POLB P06746 1/20 0.42
KDM1A O60341 1/20 0.42
GAA P10253 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPY1R P25929 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874434 1.00 EGFR (0.47) EGFRALDH1A1MAPTSMN1; SMN2ALOX12
SCHEMBL6874955 0.95 EGFR (0.54) EGFRALDH1A1MAPTSMN1; SMN2ALOX12
SCHEMBL6874938 0.95 EGFR (0.54) EGFRALDH1A1MAPTSMN1; SMN2ALOX12
SCHEMBL6874686 0.90 RAB9A (0.53) ALDH1A1MAPTSMN1; SMN2LMNAHTT
SCHEMBL6874693 0.90 RAB9A (0.53) ALDH1A1MAPTSMN1; SMN2LMNAHTT
SCHEMBL6868482 0.88 SMN1; SMN2 (0.51) ALDH1A1MAPTSMN1; SMN2LMNAHTT
SCHEMBL6868487 0.88 SMN1; SMN2 (0.51) ALDH1A1MAPTSMN1; SMN2LMNAHTT
SCHEMBL6867611 0.84 SMN1; SMN2 (0.47) ALDH1A1MAPTSMN1; SMN2LMNAMEN1
SCHEMBL6867605 0.84 SMN1; SMN2 (0.47) ALDH1A1MAPTSMN1; SMN2LMNAMEN1
SCHEMBL6878955 0.84 MCHR1 (0.43) ALDH1A1MAPTSMN1; SMN2ALOX12LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed