SCHEMBL6874607

SCHEMBL6874607

CCOc1cc(Cc2cnc(N)nc2N)cc(OS(=O)(=O)N(C)C)c1I

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.55
MEN1 O00255 1/20 0.49
SLC22A1 O15245 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
CYP2C19 P33261 1/20 0.49
BLM P54132 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6555276 0.87 DHFR (0.70) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6555506 0.85 DHFR (0.55) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6555408 0.85 DHFR (0.55) DHFR
SCHEMBL6555110 0.84 DHFR (0.53) DHFR
SCHEMBL6555188 0.84 DHFR (0.53) DHFR
SCHEMBL6554960 0.84 DHFR (0.53) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6557333 0.84 DHFR (0.53) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6555423 0.84 DHFR (0.53) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6871742 0.83 DHFR (0.52) DHFR
SCHEMBL6866298 0.83 DHFR (0.51) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6821980-B1 Substituted 5-benzyl-2,4-diaminopyrimidines BASILEA PHARMACEUTICA AG (CH) 2004-11-23 US disclosed