SCHEMBL6875101

SCHEMBL6875101

Cc1cc(CNC2CCC(Nc3nccc(N(C)C)n3)CC2)cc(C)c1O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 14/20 0.37
ADRA2A P08913 5/20 0.37
HRH1 P35367 5/20 0.37
HTR2B P41595 5/20 0.37
ADRA1A P35348 3/20 0.37
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
ACHE P22303 2/20 0.36
BACE1 P56817 1/20 0.36
MAPK14 Q16539 1/20 0.35
LCK P06239 1/20 0.35
JAK3 P52333 1/20 0.35
CNR1 P21554 1/20 0.35
KCNH2 Q12809 1/20 0.35
AURKB Q96GD4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875096 1.00 MCHR1 (0.37) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6466322 0.89 MCHR1 (0.42) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6466329 0.89 MCHR1 (0.42) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6867496 0.86 ACHE (0.44) MCHR1MAPK8MAPK9MAPK10ACHE
SCHEMBL6867477 0.86 ACHE (0.44) MCHR1MAPK8MAPK9MAPK10ACHE
SCHEMBL6873078 0.83 TSHR (0.51) MCHR1ADRA2AACHEBACE1CNR1
SCHEMBL6873081 0.83 TSHR (0.51) MCHR1ADRA2AACHEBACE1CNR1
SCHEMBL6877140 0.82 ACHE (0.42) MCHR1MAPK8MAPK9MAPK10ACHE
SCHEMBL6877144 0.82 ACHE (0.42) MCHR1MAPK8MAPK9MAPK10ACHE
SCHEMBL6876275 0.81 ACHE (0.54) HRH1HTR2BACHEBACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed