SCHEMBL6875331

SCHEMBL6875331

C[C@@H]1C(=O)N[C@@H](Cc2ccc(C(=N)N)cc2)C(=O)NCCc2ccc(F)cc2OCCN[C@@H](C2CC2)C(=O)N1C

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 20/20 0.78
CYP3A4 P08684 1/20 0.78
CYP2D6 P10635 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13552232 0.96 GHSR (0.85) GHSRCYP3A4CYP2D6
SCHEMBL13552230 0.96 GHSR (0.85) GHSRCYP3A4CYP2D6
SCHEMBL6878908 0.96 GHSR (0.85) GHSRCYP3A4CYP2D6
SCHEMBL6876644 0.96 GHSR (0.85) GHSRCYP3A4CYP2D6
SCHEMBL6875326 0.96 GHSR (0.85) GHSRCYP3A4CYP2D6
SCHEMBL6876653 0.92 GHSR (0.70) GHSRCYP3A4CYP2D6
SCHEMBL6877112 0.90 GHSR (0.75) GHSRCYP3A4CYP2D6
SCHEMBL6874019 0.90 GHSR (0.74) GHSR
SCHEMBL6874848 0.89 GHSR (0.78) GHSRCYP3A4CYP2D6
SCHEMBL804933 0.88 GHSR (1.00) GHSRCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050270-A2 MACROCYCLIC INHIBITORS OF SERINE PROTEASE ENZYMES TRANZYME PHARMA, INC. (US) 2011-04-28 WO disclosed