SCHEMBL687639

SCHEMBL687639

CSc1ccc(Cl)c(Cn2ccc(O)c(NC(=O)N[C@@H](CC(=O)O)c3ccc(C)cc3)c2=O)c1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSA P10619 8/20 0.36
PTGER3 P43115 2/20 0.36
CYP26A1 O43174 4/20 0.35
KEAP1 Q14145 2/20 0.33
NFE2L2 Q16236 2/20 0.33
ITGB1 P05556 2/20 0.33
ITGA4 P13612 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687691 0.89 PTGER3 (0.41) CTSAPTGER3CYP26A1
SCHEMBL688035 0.87 CTSA (0.41) CTSAPTGER3KDM4EPOLBMAPT
SCHEMBL688155 0.87 PTGER3 (0.49) CTSAPTGER3KDM4EPOLBMAPT
SCHEMBL688040 0.87 PTGER3 (0.49) CTSAPTGER3KDM4EPOLBMAPT
SCHEMBL687149 0.86 CTSA (0.47) CTSAPTGER3CYP26A1MAPT
SCHEMBL688150 0.86 ITGB1 (0.38) CTSAPTGER3CYP26A1KEAP1NFE2L2
SCHEMBL688248 0.85 POLB (0.39) CTSACYP26A1KEAP1NFE2L2ITGB1
SCHEMBL687628 0.85 KMT2A (0.42) CTSAPTGER3CYP26A1KDM4EMAPT
SCHEMBL687906 0.84 PTGER3 (0.47) CTSAPTGER3ITGB1ITGA4KDM4E
SCHEMBL688413 0.84 POLB (0.40) CTSACYP26A1KEAP1NFE2L2ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed