SCHEMBL6876584

SCHEMBL6876584

CC(C)S(=O)(=O)c1csc(C(=O)N[C@H]2CC[C@@H](Nc3nccc(N(C)C)n3)CC2)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
CDK7 P50613 2/20 0.43
CDK9 P50750 2/20 0.43
MCHR1 Q99705 15/20 0.42
ADRA2A P08913 7/20 0.42
HRH1 P35367 7/20 0.42
HTR2B P41595 6/20 0.42
ADRA1A P35348 4/20 0.42
POLB P06746 1/20 0.42
CNR1 P21554 1/20 0.38
KCNH2 Q12809 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876589 1.00 KDM4E (0.46) KDM4EGAACDK7CDK9MCHR1
SCHEMBL6880618 0.90 MCHR1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6880622 0.90 MCHR1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6467272 0.82 MCHR1 (0.40) CDK7CDK9MCHR1ADRA2AHRH1
SCHEMBL6467267 0.82 MCHR1 (0.40) CDK7CDK9MCHR1ADRA2AHRH1
SCHEMBL13793609 0.80 MCHR1 (0.58) KDM4EGAAMCHR1ADRA2AHRH1
SCHEMBL6868087 0.79 KDM4E (0.44) KDM4EGAAMCHR1ADRA2AHRH1
SCHEMBL6868092 0.79 KDM4E (0.44) KDM4EGAAMCHR1ADRA2AHRH1
SCHEMBL6880308 0.79 MCHR1 (0.48) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6880312 0.79 MCHR1 (0.48) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed