SCHEMBL687660

SCHEMBL687660

O=C(O)C[C@H](NC(=O)Nc1c(O)ccn(Cc2ccccc2Cl)c1=O)c1ccc2c(c1)OCO2

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.44
ITGAV P06756 6/20 0.44
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 2/20 0.41
ITGA2B P08514 7/20 0.41
PTGER3 P43115 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687498 0.96 ALDH1A1 (0.42) ITGB3ITGAVKMT2AMEN1POLB
SCHEMBL687672 0.88 CYP26A1 (0.43) ALDH1A1PTGER3
SCHEMBL687418 0.87 PTGER3 (0.46) ALDH1A1PTGER3
SCHEMBL687428 0.87 PTGER3 (0.56) ITGB3ITGAVKMT2AMEN1ALDH1A1
SCHEMBL687886 0.87 PTGER3 (0.56) ITGB3ITGAVKMT2AMEN1ALDH1A1
SCHEMBL687411 0.87 PTGER3 (0.42) ALDH1A1PTGER3
SCHEMBL687520 0.86 PTGER3 (0.42) KMT2APOLBALDH1A1PTGER3
SCHEMBL688004 0.86 PTGER3 (0.44) KMT2AMEN1ALDH1A1PTGER3
SCHEMBL687155 0.86 PTGER3 (0.44) ALDH1A1PTGER3
SCHEMBL687771 0.86 PTGER3 (0.45) ALDH1A1PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1176956-B1 CARBOXYLIC ACID DERIVATIVES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed