SCHEMBL6876607

SCHEMBL6876607

CN(C)c1cc(NC2CCC(NC(=O)Nc3ccccc3C(F)(F)F)CC2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.47
MCHR1 Q99705 8/20 0.45
ADRA2A P08913 6/20 0.45
EPHX2 P34913 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
HTR2B P41595 1/20 0.41
NPY5R Q15761 1/20 0.41
EPHX1 P07099 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876600 1.00 ACP1 (0.47) ACP1MCHR1ADRA2AEPHX2MEN1
SCHEMBL6878561 0.92 P2RY1 (0.43) MCHR1ADRA2AKDM4EHTR1AADRA1A
SCHEMBL6878565 0.92 P2RY1 (0.43) MCHR1ADRA2AKDM4EHTR1AADRA1A
SCHEMBL6868426 0.91 MCHR1 (0.44) ACP1MCHR1ADRA2AKDM4ETRPV1
SCHEMBL6872387 0.91 MCHR1 (0.46) ACP1MCHR1ADRA2AHTR1AADRA1A
SCHEMBL6872384 0.91 MCHR1 (0.46) ACP1MCHR1ADRA2AHTR1AADRA1A
SCHEMBL6868434 0.91 MCHR1 (0.44) ACP1MCHR1ADRA2AKDM4ETRPV1
SCHEMBL6867920 0.90 ACP1 (0.44) ACP1MCHR1ADRA2AEPHX2MEN1
SCHEMBL6867914 0.90 ACP1 (0.44) ACP1MCHR1ADRA2AEPHX2MEN1
SCHEMBL6868474 0.88 MCHR1 (0.44) ACP1MCHR1ADRA2AEPHX2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed