SCHEMBL6876802

SCHEMBL6876802

COC(=O)c1cccc(NC(=S)NC2CCC(Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
LMNA P02545 2/20 0.47
RAB9A P51151 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MCHR1 Q99705 7/20 0.43
ADRA2A P08913 6/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
HTR2B P41595 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 3/20 0.42
ALDH1A1 P00352 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876788 1.00 NPC1 (0.47) NPC1LMNARAB9ANFKB1NFKB2
SCHEMBL6879594 0.92 NPC1 (0.57) NPC1LMNASMN1; SMN2MCHR1ADRA2A
SCHEMBL6879588 0.92 NPC1 (0.57) NPC1LMNASMN1; SMN2MCHR1ADRA2A
SCHEMBL6868594 0.92 MAPT (0.47) NPC1LMNARAB9ASMN1; SMN2MCHR1
SCHEMBL6867921 0.92 EPHX2 (0.49) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL6867915 0.92 EPHX2 (0.49) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL6875046 0.92 NPC1 (0.48) NPC1LMNASMN1; SMN2MCHR1ADRA2A
SCHEMBL6875057 0.92 NPC1 (0.48) NPC1LMNASMN1; SMN2MCHR1ADRA2A
SCHEMBL6875557 0.90 MEN1 (0.56) NPC1SMN1; SMN2MCHR1ADRA2AADRA1A
SCHEMBL6875563 0.90 MEN1 (0.56) NPC1SMN1; SMN2MCHR1ADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed