SCHEMBL6879588

SCHEMBL6879588

CC(=O)c1cccc(NC(=S)N[C@H]2CC[C@@H](Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
LMNA P02545 1/20 0.57
MCHR1 Q99705 9/20 0.45
ADRA2A P08913 8/20 0.45
ADRA1A P35348 1/20 0.45
HRH1 P35367 1/20 0.45
HTR2B P41595 1/20 0.45
PKM P14618 1/20 0.44
ALOX15 P16050 1/20 0.44
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX12 P18054 1/20 0.41
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879594 1.00 NPC1 (0.57) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6875057 0.94 NPC1 (0.48) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6875046 0.94 NPC1 (0.48) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6876788 0.92 NPC1 (0.47) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6876802 0.92 NPC1 (0.47) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6880607 0.91 PKM (0.55) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6880600 0.91 PKM (0.55) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6867093 0.90 MEN1 (0.45) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6867086 0.90 MEN1 (0.45) NPC1LMNAMCHR1ADRA2AADRA1A
SCHEMBL6868594 0.89 MAPT (0.47) NPC1LMNAMCHR1ADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed