SCHEMBL6877102

SCHEMBL6877102

CN(C)c1nc(NC2CCC(NC(=O)Nc3ccc(F)c(F)c3)CC2)nc2c1CCCC2

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MCHR1 Q99705 14/20 0.52
ADRA2A P08913 7/20 0.49
HRH1 P35367 4/20 0.49
HTR2B P41595 4/20 0.49
ADRA1A P35348 3/20 0.49
HTR1A P08908 1/20 0.49
NPY5R Q15761 1/20 0.49
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
KMT2A Q03164 1/20 0.45
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
EPHX2 P34913 1/20 0.41
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877094 1.00 NPC1 (0.53) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6878058 0.92 MEN1 (0.58) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6878062 0.92 MEN1 (0.58) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6879056 0.90 MCHR1 (0.44) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6879059 0.90 MCHR1 (0.44) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6465036 0.90 MCHR1 (0.51) NPC1RAB9AMCHR1ADRA2AHRH1
SCHEMBL6465026 0.90 MCHR1 (0.51) NPC1RAB9AMCHR1ADRA2AHRH1
SCHEMBL6868342 0.89 MEN1 (0.44) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6868349 0.89 MEN1 (0.44) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A
SCHEMBL6868970 0.89 MCHR1 (0.54) NPC1RAB9ASMN1; SMN2MCHR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed