SCHEMBL6877104

SCHEMBL6877104

CCc1cccc(CC)c1NC(=O)N[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 11/20 0.43
KDR P35968 1/20 0.42
AURKB Q96GD4 2/20 0.41
KMT2A Q03164 1/20 0.41
ADRA2A P08913 4/20 0.40
HRH1 P35367 4/20 0.40
HTR2B P41595 4/20 0.40
ADRA1A P35348 2/20 0.40
CYP2C9 P11712 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39
EPHX1 P07099 1/20 0.38
TP53 P04637 1/20 0.38
CNR1 P21554 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877107 1.00 MCHR1 (0.43) MCHR1KDRAURKBKMT2AADRA2A
SCHEMBL6880721 0.94 TP53 (0.46) MCHR1KDRAURKBADRA2AHRH1
SCHEMBL6880714 0.94 TP53 (0.46) MCHR1KDRAURKBADRA2AHRH1
SCHEMBL6868958 0.92 EPHX2 (0.42) MCHR1KDRAURKBKMT2AADRA2A
SCHEMBL6868955 0.92 EPHX2 (0.42) MCHR1KDRAURKBKMT2AADRA2A
SCHEMBL6874218 0.89 MCHR1 (0.41) MCHR1KMT2AADRA2AHRH1HTR2B
SCHEMBL6877414 0.89 KMT2A (0.56) MCHR1KDRAURKBKMT2AADRA2A
SCHEMBL6874211 0.89 MCHR1 (0.41) MCHR1KMT2AADRA2AHRH1HTR2B
SCHEMBL6877409 0.89 KMT2A (0.56) MCHR1KDRAURKBKMT2AADRA2A
SCHEMBL6463172 0.88 MCHR1 (0.43) MCHR1KDRADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed