SCHEMBL6868955

SCHEMBL6868955

CCc1cccc(C(C)C)c1NC(=O)N[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
MCHR1 Q99705 8/20 0.39
KDR P35968 1/20 0.39
AURKB Q96GD4 1/20 0.38
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
MAPK10 P53779 2/20 0.37
ADRA2A P08913 2/20 0.36
ADRA1A P35348 2/20 0.36
HRH1 P35367 2/20 0.36
HTR2B P41595 2/20 0.36
KMT2A Q03164 1/20 0.36
NMBR P28336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868958 1.00 EPHX2 (0.42) EPHX2MCHR1KDRAURKBMAPK8
SCHEMBL6877107 0.92 MCHR1 (0.43) MCHR1KDRAURKBMAPK8MAPK9
SCHEMBL6877104 0.92 MCHR1 (0.43) MCHR1KDRAURKBMAPK8MAPK9
SCHEMBL6873242 0.90 MCHR1 (0.37) MCHR1MAPK8MAPK9MAPK10ADRA2A
SCHEMBL6873247 0.90 MCHR1 (0.37) MCHR1MAPK8MAPK9MAPK10ADRA2A
SCHEMBL6457210 0.90 MCHR1 (0.40) EPHX2MCHR1ADRA2AADRA1AHRH1
SCHEMBL6457203 0.90 MCHR1 (0.40) EPHX2MCHR1ADRA2AADRA1AHRH1
SCHEMBL6875772 0.89 EPHX1 (0.44) EPHX2MCHR1KDRAURKBADRA2A
SCHEMBL6875782 0.89 EPHX1 (0.44) EPHX2MCHR1KDRAURKBADRA2A
SCHEMBL6880721 0.88 TP53 (0.46) EPHX2MCHR1KDRAURKBADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed