SCHEMBL687714

SCHEMBL687714

CCC(C(=O)O)[C@H](O)CC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.42
CHRM1 P11229 1/20 0.42
AKR1A1 P14550 1/20 0.42
CHRM3 P20309 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
ADRA1A P35348 1/20 0.42
HRH1 P35367 1/20 0.42
DRD3 P35462 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
TP53 P04637 1/20 0.38
CA2 P00918 1/20 0.36
MAPK1 P28482 1/20 0.36
GPR84 Q9NQS5 3/20 0.34
SLC1A3 P43003 2/20 0.34
SLC1A2 P43004 2/20 0.34
SLC1A1 P43005 2/20 0.34
FFAR1 O14842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837519 1.00 TDP1 (0.42) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL3064781 0.84 PDE4A (0.44) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL27677822 0.84 OR51E2 (0.42) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL1895730 0.84 PDE4A (0.44) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL3064788 0.84 PDE4A (0.44) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL3073651 0.84 PDE4A (0.44) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL5489376 0.82 PTGS1 (0.37) TDP1TP53
SCHEMBL13986496 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL9636422 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A
SCHEMBL1000793 0.82 TDP1 (0.48) TDP1CHRM1AKR1A1CHRM3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871782-B1 DIPHOSPHINES AND METAL COMPLEXES UMICORE AG & CO KG (DE) 2012-02-29 EP disclosed
EP-1904640-B1 ASYMMETRIC REDUCTION OF 1,1,1-TRIFLUOROACETONE HOFFMANN LA ROCHE (CH) 2009-08-19 EP disclosed
EP-1904640-A2 ASYMMETRIC REDUCTION OF 1,1,1-TRIFLUOROACETONE F. Hoffmann-Roche AG (CH) 2008-04-02 EP disclosed
US-7196234-B2 Asymmetric reduction of 1,1,1-trifluoroacetone HOFFMAN-LA ROCHE INC. (US) 2007-03-27 US disclosed
WO-2007006650-A2 ASYMMETRIC REDUCTION OF 1,1,1-TRIFLUOROACETONE F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed
US-20070009999-A1 Asymmetric reduction of 1,1,1-trifluoroacetone HOFFMANN-LA ROCHE INC. 2007-01-11 US disclosed