SCHEMBL6877259

SCHEMBL6877259

Cc1cc(Cl)ccc1NC(=S)N[C@H]1CC[C@@H](Nc2cc(N(C)C)c3ccccc3n2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
KDR P35968 1/20 0.43
NPC1 O15118 2/20 0.43
THRB P10828 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MCHR1 Q99705 2/20 0.42
ADRA2A P08913 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NOX1 Q9Y5S8 1/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALPL P05186 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877266 1.00 SMN1; SMN2 (0.44) SMN1; SMN2KDRNPC1THRBRAB9A
SCHEMBL6876734 0.92 MEN1 (0.51) SMN1; SMN2NPC1RAB9ALMNAKDM4E
SCHEMBL6876725 0.92 MEN1 (0.51) SMN1; SMN2NPC1RAB9ALMNAKDM4E
SCHEMBL6877176 0.91 TP53 (0.47) SMN1; SMN2NPC1RAB9ALMNAKDM4E
SCHEMBL6877168 0.91 TP53 (0.47) SMN1; SMN2NPC1RAB9ALMNAKDM4E
SCHEMBL6880440 0.89 KDR (0.51) SMN1; SMN2KDRNPC1RAB9ALMNA
SCHEMBL6873091 0.89 KDM4E (0.43) SMN1; SMN2LMNAKDM4EMCHR1ADRA2A
SCHEMBL6458568 0.89 SMN1; SMN2 (0.43) SMN1; SMN2LMNAKDM4EMCHR1ADRA2A
SCHEMBL6880443 0.89 KDR (0.51) SMN1; SMN2KDRNPC1RAB9ALMNA
SCHEMBL6873096 0.89 KDM4E (0.43) SMN1; SMN2LMNAKDM4EMCHR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed