SCHEMBL6877366

SCHEMBL6877366

CN(C)c1cc(N[C@H]2CC[C@@H](NC(=O)c3cccc(Oc4ccccc4)c3)CC2)nc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.61
PKM P14618 1/20 0.56
MCHR1 Q99705 16/20 0.54
ADRA2A P08913 12/20 0.54
ADRA1A P35348 2/20 0.49
HRH1 P35367 2/20 0.49
HTR2B P41595 2/20 0.49
HTR1A P08908 1/20 0.49
NPY5R Q15761 1/20 0.49
CCR3 P51677 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877371 1.00 NPC1 (0.61) NPC1PKMMCHR1ADRA2AADRA1A
SCHEMBL6465595 0.93 MCHR1 (0.61) NPC1MCHR1ADRA2AADRA1AHRH1
SCHEMBL6465599 0.93 MCHR1 (0.61) NPC1MCHR1ADRA2AADRA1AHRH1
SCHEMBL6457452 0.89 MCHR1 (0.55) NPC1PKMMCHR1ADRA2AADRA1A
SCHEMBL6457460 0.89 MCHR1 (0.55) NPC1PKMMCHR1ADRA2AADRA1A
SCHEMBL6879865 0.89 MCHR1 (0.57) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6879862 0.89 MCHR1 (0.57) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6873154 0.89 MCHR1 (0.58) NPC1MCHR1ADRA2AADRA1AHRH1
SCHEMBL6873148 0.89 MCHR1 (0.58) NPC1MCHR1ADRA2AADRA1AHRH1
SCHEMBL6455557 0.88 MCHR1 (0.70) NPC1MCHR1ADRA2AADRA1AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed