SCHEMBL6877776

SCHEMBL6877776

COc1ccc(OC)c(CNC2CCC(Nc3cc(N(C)C)c4ccccc4n3)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 12/20 0.50
ADRA2A P08913 1/20 0.43
TACR1 P25103 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MDM2 Q00987 1/20 0.43
APP P05067 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TP53 P04637 2/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877772 1.00 MCHR1 (0.50) MCHR1ADRA2ATACR1ALDH1A1MDM2
SCHEMBL6874467 0.93 MCHR1 (0.50) MCHR1ADRA2AALDH1A1MEN1KMT2A
SCHEMBL6874473 0.93 MCHR1 (0.50) MCHR1ADRA2AALDH1A1MEN1KMT2A
SCHEMBL6879011 0.91 MCHR1 (0.51) MCHR1ADRA2AALDH1A1APPBCHE
SCHEMBL6879016 0.91 MCHR1 (0.51) MCHR1ADRA2AALDH1A1APPBCHE
SCHEMBL6873885 0.89 MCHR1 (0.46) MCHR1ADRA2AALDH1A1MDM2APP
SCHEMBL6873877 0.89 MCHR1 (0.46) MCHR1ADRA2AALDH1A1MDM2APP
SCHEMBL6873630 0.89 MCHR1 (0.51) MCHR1ADRA2AAPPBCHEACHE
SCHEMBL6873635 0.89 MCHR1 (0.51) MCHR1ADRA2AAPPBCHEACHE
SCHEMBL6873798 0.88 SIGMAR1 (0.54) MCHR1ADRA2AMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed