SCHEMBL687791

SCHEMBL687791

COc1ccc(-c2ccc([C@H](CC(=O)O)NC(=O)Nc3c(O)c(C)cn(Cc4ccccc4Cl)c3=O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 5/20 0.43
CTSA P10619 7/20 0.42
ALDH1A1 P00352 2/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CNR2 P34972 1/20 0.37
EDNRB P24530 1/20 0.37
UTS2R Q9UKP6 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686842 0.98 PTGER3 (0.45) PTGER3CTSAALDH1A1THRBHPGD
SCHEMBL687923 0.94 PTGER3 (0.41) PTGER3CTSACNR2UTS2R
SCHEMBL686938 0.91 PTGER3 (0.47) PTGER3CTSAALDH1A1THRBHPGD
SCHEMBL688053 0.90 PTGER3 (0.43) PTGER3CTSAALDH1A1RXFP1CNR2
SCHEMBL688669 0.90 PTGER3 (0.42) PTGER3CTSACNR2
SCHEMBL687527 0.90 ITGB1 (0.42) PTGER3CTSATHRBCNR2
SCHEMBL686799 0.90 PTGER3 (0.51) PTGER3CTSATHRBCNR2SMN1; SMN2
SCHEMBL686896 0.89 PTGER3 (0.44) PTGER3CTSACNR2
SCHEMBL688284 0.89 PTGER3 (0.43) PTGER3CTSAALDH1A1CNR2SMN1; SMN2
SCHEMBL29371834 0.89 PTGER3 (0.44) PTGER3CTSACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed