SCHEMBL686938

SCHEMBL686938

COc1ccc2cc([C@H](CC(=O)O)NC(=O)Nc3c(O)c(C)cn(Cc4ccccc4Cl)c3=O)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 8/20 0.47
CTSA P10619 3/20 0.39
GCGR P47871 1/20 0.38
LCK P06239 1/20 0.37
P2RX7 Q99572 2/20 0.37
ALDH1A1 P00352 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CYP26A1 O43174 1/20 0.36
CNR2 P34972 1/20 0.36
SLC22A12 Q96S37 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686799 0.93 PTGER3 (0.51) PTGER3CTSATHRBCNR2SLC22A12
SCHEMBL686846 0.93 PTGER3 (0.41) PTGER3CTSAALDH1A1CYP26A1CNR2
SCHEMBL686842 0.93 PTGER3 (0.45) PTGER3CTSALCKALDH1A1THRB
SCHEMBL687791 0.91 PTGER3 (0.43) PTGER3CTSAALDH1A1THRBHPGD
SCHEMBL687310 0.90 CTSA (0.39) PTGER3CTSAGCGRALDH1A1THRB
SCHEMBL688343 0.89 PTGER3 (0.43) PTGER3CTSAP2RX7RXFP1CNR2
SCHEMBL688233 0.89 PTGER3 (0.43) PTGER3CTSAP2RX7RXFP1CYP26A1
SCHEMBL688170 0.88 PTGER3 (0.41) PTGER3ALDH1A1RXFP1CYP26A1CNR2
SCHEMBL687540 0.88 PTGER3 (0.48) PTGER3CTSAGCGRLCKALDH1A1
SCHEMBL688406 0.88 PTGER3 (0.48) PTGER3CTSAGCGRLCKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed