SCHEMBL6877945

SCHEMBL6877945

CCOc1ccc2ccccc2c1C(=O)N[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
TP53 P04637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CXCR5 P32302 1/20 0.44
ABCB11 O95342 1/20 0.42
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MCHR1 Q99705 10/20 0.41
HIF1A Q16665 1/20 0.41
HCRTR1 O43613 3/20 0.41
HCRTR2 O43614 3/20 0.41
ADRA2A P08913 4/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877953 1.00 ALDH1A1 (0.45) ALDH1A1TP53L3MBTL1CXCR5ABCB11
SCHEMBL6874502 0.85 MCHR1 (0.48) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6874497 0.85 MCHR1 (0.48) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6877203 0.84 USP2 (0.48) ALDH1A1MCHR1HCRTR1HCRTR2
SCHEMBL6877198 0.84 USP2 (0.48) ALDH1A1MCHR1HCRTR1HCRTR2
SCHEMBL13793521 0.83 MCHR1 (0.61) CXCR5MCHR1ADRA2AADRA1AHRH1
SCHEMBL6877485 0.81 MCHR1 (0.52) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6877476 0.81 MCHR1 (0.52) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6877756 0.80 MCHR1 (0.45) CXCR5MCHR1ADRA2AADRA1AHRH1
SCHEMBL6877757 0.80 MCHR1 (0.45) CXCR5MCHR1ADRA2AADRA1AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed