SCHEMBL6878124

SCHEMBL6878124

CN(C)c1ccnc(NC2CCC(NC(=O)c3cc4ccccc4s3)CC2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
CHRNA7 P36544 4/20 0.47
HTR3A P46098 3/20 0.47
MCHR1 Q99705 9/20 0.46
MEN1 O00255 1/20 0.46
ADRA2A P08913 3/20 0.45
HRH1 P35367 3/20 0.45
HTR2B P41595 3/20 0.45
ADRA1A P35348 2/20 0.45
OPRM1 P35372 1/20 0.45
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878117 1.00 RAB9A (0.48) RAB9AKMT2ANPC1CHRNA7HTR3A
SCHEMBL6460134 0.83 MCHR1 (0.47) RAB9AKMT2AMCHR1MEN1ADRA2A
SCHEMBL6463225 0.83 MCHR1 (0.47) RAB9AKMT2AMCHR1MEN1ADRA2A
SCHEMBL6879782 0.82 RAB9A (0.51) RAB9AKMT2ANPC1MCHR1MEN1
SCHEMBL6879777 0.82 RAB9A (0.51) RAB9AKMT2ANPC1MCHR1MEN1
SCHEMBL6878847 0.81 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6878850 0.81 MCHR1 (0.58) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6874497 0.81 MCHR1 (0.48) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6877882 0.81 MCHR1 (0.59) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6874502 0.81 MCHR1 (0.48) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed