SCHEMBL6878376

SCHEMBL6878376

OCC=C(F)c1ccc(-c2ccncn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.43
HDAC4 P56524 1/20 0.36
ROCK1 Q13464 2/20 0.35
GSK3B P49841 2/20 0.35
ROCK2 O75116 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
PRKCG P05129 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
MAPK1 P28482 1/20 0.35
GSK3A P49840 1/20 0.35
PRKX P51817 1/20 0.35
PRKCD Q05655 1/20 0.35
PRKG1 Q13976 1/20 0.35
PKN2 Q16513 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
SGK2 Q9HBY8 1/20 0.35
MAPK14 Q16539 4/20 0.34
MAPK10 P53779 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878374 1.00 CYP2D6 (0.43) CYP2D6HDAC4ROCK1GSK3BROCK2
SCHEMBL6878371 1.00 CYP2D6 (0.43) CYP2D6HDAC4ROCK1GSK3BROCK2
SCHEMBL6852058 0.81 CYP2D6 (0.42) CYP2D6HDAC4ROCK1GSK3BROCK2
SCHEMBL6852059 0.81 CYP2D6 (0.42) CYP2D6HDAC4ROCK1GSK3BROCK2
SCHEMBL6879912 0.80 HDAC1 (0.42) ROCK1GSK3BROCK2PRKCGPRKACA
SCHEMBL6879909 0.80 HDAC1 (0.42) ROCK1GSK3BROCK2PRKCGPRKACA
SCHEMBL6879903 0.80 HDAC1 (0.42) ROCK1GSK3BROCK2PRKCGPRKACA
SCHEMBL6869722 0.80 TRPV1 (0.43) CYP2D6CYP2C9
SCHEMBL6869718 0.80 TRPV1 (0.43) CYP2D6CYP2C9
SCHEMBL6869713 0.80 TRPV1 (0.43) CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed